Name
AS-8351,KDM5B histone demethylase inhibitor
Size
25 mg
Catalog number
SIH-558-25MG
Price
470 EUR
More details
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Research Area(s)
Stem Cells
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Category
Small Molecules
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Product Type
Inhibitor
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CAS No.
796-42-9
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MolecularFormula
C17H13N3O2
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Molecular Weight
291.3
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Purity
>98% (TLC); NMR (Conforms)
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Solubility
May be dissolved in DMSO (45 mg/ml); or ethanol (10 mg/ml, warm); or DMF (30 mg/ml)
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Appearance
Yellow powder
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Storage Temperature
-20°C
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Shipping Temperature
Blue Ice or 4ºC
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Description
Tissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.